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GPCR Products

Ready-to-Assay Cell Lines and Membranes

We are continually striving to develop innovative products for GPCR research. Our Ready-to-Assay product line accelerates GPCR drug discovery by providing convenience for routine drug assays.

» View Product Listing - Ready-to-Assay Cell Lines
» View Product Listing - Ready-to-Assay Membranes

Ready-to-Assay GPCR Calcium-Optimized Cells

• Cell-based assays within 24 hrs from start to finish
• Cryopreserved version of ChemiScreen Calcium-Optimized GPCR Cell Lines
• High cellular viability and assay signal
• Preserved pharmacology
• Available in bulk quantities

Comparison of Potency and Efficacy of Ready-to-Assay GPCR Calcium-Optimized Cells Versus Traditional Continuously Passaged ChemiScreen GPCR Calcium-Optimized Stable Cell Lines By Ca²⁺ Flux Assay

Product Listing

Class	Ligand Type	GPCR Family	GPCR Target (Human unless noted)	Cell Line Host	Ready-to-Assay Cells Catalogue Number
A	non-peptide	Adrenergic	alpha1a	Chem-1	HTS087F	Coming soon
A	non-peptide	Adrenergic	alpha2a	Chem-1	HTS096F	Coming soon
A	non-peptide	Adrenergic	alpha2b	Chem-1	HTS156F	New
A	non-peptide	Adrenergic	beta1	Chem-1	HTS104F	New
A	non-peptide	Adrenergic	beta2	Chem-2	HTS073F	New
A	non-peptide	Adrenergic	beta3	Chem-10	HTS159F	New
A	non-peptide	Cannabinoid	CB1	Chem-1	HTS019F	New
A	non-peptide	Cannabinoid	CB2	Chem-4	HTS020F	New
A	peptide	Chemoattractant	ChemR23	Chem-1	HTS071F	Coming soon
A	peptide	Chemokine	CCR1	Chem-1	HTS005F
A	peptide	Chemokine	CCR2B	Chem-1	HTS007F
A	peptide	Chemokine	CCR4	Chem-5	HTS009F
A	peptide	Chemokine	CCR5, rhesus macaque	Chem-1	HTS010F	New
A	peptide	Chemokine	CCR9	Chem-1	HTS036F
A	peptide	Chemokine	CXCR1	Chem-1	HTS001F
A	peptide	Chemokine	CXCR2	Chem-1	HTS002F
A	peptide	Chemokine	CXCR3	Chem-1	HTS003F
A	peptide	Chemokine	CXCR4	Chem-1	HTS004F
B	peptide	CRF Receptor	CRF1	Chem-1	HTS023F
B	peptide	CRF Receptor	CRF2	Chem-1	HTS024F
A	non-peptide	Free Fatty Acid	GPR40	Chem-1	HTS038F	Coming Soon
A	non-peptide	Free Fatty Acid	GPR41	Chem-4	HTS135F	New
A	non-peptide	Free Fatty Acid	GPR43	Chem-1	HTS063F	New
C	non-peptide	GABAB	GABAB1b	Chem-1	HTS119F	Coming soon
B	peptide	Glucagon	GIP	Chem-9	HTS134F	New
B	peptide	Glucagon	glucagon	Chem-1	HTS112F	Coming soon
B	peptide	Glucagon	secretin receptor	Chem-1	HTS174F	New
C	non-peptide	Glutamate (metabotropic)	mGlu2	Chem-1	HTS146F
A	non-peptide	Leukotriene	BLT1	Chem-1	HTS042F
A	non-peptide	Leukotriene	CysLT1	Chem-1	HTS061F
A	non-peptide	Lysophospholipid	LPA3	Chem-1	HTS130F
A	non-peptide	Lysophospholipid	S1P1	Chem-4	HTS176F	New
A	non-peptide	Lysophospholipid	S1P2	Chem-1	HTS078F
A	non-peptide	Lysophospholipid	S1P3	Chem-1	HTS097F
A	non-peptide	Lysophospholipid	S1P4	Chem-5	HTS192F
A	peptide	Neuropeptide Y	Y2	Chem-1	HTS066F
A	peptide	Neurotensin	NTR1	Chem-1	HTS034F
A	peptide	N-formylpeptide	FPRL1	Chem-1	HTS056F
A	peptide	Orexin	OX1	Chem-1	HTS175F
A	peptide	Orexin	OX2	Chem-1	HTS045F
A	non-peptide	Prostanoid	DP	Chem-1	HTS091F
A	non-peptide	Prostanoid	EP1	Chem-1	HTS099F
A	non-peptide	Prostanoid	EP2	Chem-9	HTS185F
A	non-peptide	Prostanoid	EP3	Chem-1	HTS092F
A	non-peptide	Prostanoid	EP4	Chem-1	HTS142F
A	non-peptide	Prostanoid	FP	Chem-1	HTS093F
A	non-peptide	Prostanoid	IP1	Chem-1	HTS131F	New
A	non-peptide	Prostanoid	TP	Chem-1	HTS081F
B	peptide	PTH receptor	PTH1	Chem-1	HTS030F
B	peptide	PTH receptor	PTH2	Chem-1	HTS173	New
A	peptide	Vasopressin	V1A	Chem-1	HTS059F	Coming soon
B	peptide	VIP/PACAP	VPAC1	Chem-1	HTS043F	New

Ready-to-Assay Pre-Plated Membranes

• Millipore GPCR membranes pre-aliquoted onto assay plates
• Reduced steps compared to traditional filtration
• Single plate for both assay & filtration
• Amenable to automation
• High signal-to-noise
• Available in bulk quantities

Comparison of Affinity and Total Binding of Ready-to-Assay Pre-plated GPCR Membrane Preparations Versus Conventional Filtration Assays Using ChemiScreen GPCR Membrane Preparations.

Product Listing

Class	Ligand Type	GPCR Family	GPCR Target (Human unless noted)	Membrane host	Ready-to-Assay Pre-plated membranes
A	non-peptide	Adenosine	A3	Chem-3	HTS052P	Coming Soon
A	non-peptide	Adrenergic	alpha1A	Chem-1	HTS087P	New
A	non-peptide	Adrenergic	beta 1	Chem-1	HTS104P	New
A	non-peptide	Adrenergic	beta 2	Chem-2	HTS073P	New
A	non-peptide	Adrenergic	beta 3	Chem-1	HTS159P	New
A	non-peptide	Prostanoid	CRTH2	Chem-1	HTS031P
A	non-peptide	Prostanoid	EP2	Chem-1	HTS185P	New
A	non-peptide	Prostanoid	EP3	Chem-1	HTS092P
A	non-peptide	Prostanoid	EP4	Chem-1	HTS142P
A	non-peptide	Prostanoid	TP	Chem-1	HTS081P
A	non-peptide	Prostanoid	CRTH2, DP, EP3, EP4, TP array	Chem-1	HTS900PA

Featured Products

• Mouse Soluble Cytokine Receptor Panel
  (13 analytes)
• Human Cytokine/Chemokine Panel
• Mouse Cytokine/Chemokine Panel
• Non-Human Primate Cytokine/Chemokine Panel
• Human Apoptosis Cell Signaling Panel
• cAMP 384-well Plate Kit
• cGMP 384-well Plate Kit
• BioForm Technology for Tyrosine Kinases
• Lipid Kinases

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• Primary
• Secondary

Find Primary Antibodies

Enter a keyword and/or search criteria below. Or you may also use selections below to browse specific antibodies for your needs.

Keyword Gene Symbol UniProt Number Entrez Gene Number

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Find Secondary Antibodies

Select the host, conjugate, and species, and then press Search to find the secondary antibodies for your research needs.